SCHEMBL11043870

SCHEMBL11043870

C[C@@H]1C(=O)c2ccccc2O[C@H]1c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.56
RET P07949 1/20 0.50
KDR P35968 1/20 0.50
CYP19A1 P11511 5/20 0.49
MAOB P27338 4/20 0.49
ADORA3 P0DMS8 2/20 0.49
KDM4E B2RXH2 1/20 0.49
AR P10275 1/20 0.49
HSD17B10 Q99714 1/20 0.49
MAPT P10636 3/20 0.42
CYP3A4 P08684 2/20 0.42
MAPK1 P28482 2/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
HTR2B P41595 1/20 0.42
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
DNMT3B Q9UBC3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5579742 1.00 ESR1 (0.56) ESR1RETKDRCYP19A1MAOB
SCHEMBL7522409 0.88 ESR1 (0.56) ESR1RETKDRCYP19A1MAOB
SCHEMBL5579748 0.88 ESR1 (0.56) ESR1RETKDRCYP19A1MAOB
SCHEMBL24227321 0.81 ESR1 (0.68) ESR1CYP19A1MAOBAR
SCHEMBL4360680 0.81 ESR1 (0.86) ESR1CYP19A1MAOBADORA3KDM4E
SCHEMBL28186146 0.80 RET (0.51) RETKDRCYP19A1MAOBADORA3
SCHEMBL16376660 0.80 ESR1 (0.55) ESR1RETKDRCYP19A1MAOB
SCHEMBL92288 0.79 ESR1 (0.45) ESR1RETKDRCYP19A1MAOB
SCHEMBL9434848 0.79 ESR1 (0.45) ESR1RETKDRCYP19A1MAOB
SCHEMBL8702376 0.79 ESR1 (0.45) ESR1RETKDRCYP19A1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0025599-B1 BENZOPYRAN COMPOUNDS, USEFUL AS CHEMOTHERAPEUTIC AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1984-12-19 EP disclosed
US-4452991-A OR BENZO(B)INDENO (2,1-E) PYRANS OR BENZO(C)XANTHENES BATCHELOR JOHN F (GB) 1984-06-05 US disclosed
EP-0025599-A1 Benzopyran compounds, useful as chemotherapeutic agents THE WELLCOME FOUNDATION LIMITED (GB) 1981-03-25 EP disclosed