SCHEMBL11044112

SCHEMBL11044112

COc1ccc(CC(F)(Cc2c[nH]nn2)c2ccc(Cl)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
MAPT P10636 4/20 0.36
KDR P35968 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
NPBWR1 P48145 1/20 0.35
CXCR3 P49682 1/20 0.35
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
ALOX5 P09917 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11050458 0.88 SLC6A2 (0.33) LMNASMN1; SMN2ALDH1A1GAA
SCHEMBL11046338 0.86 CYP19A1 (0.37) HTTKMT2ASMN1; SMN2MAPTCXCR3
SCHEMBL11046622 0.86 LMNA (0.39) LMNAHTTNPSR1MEN1KMT2A
SCHEMBL11043557 0.86 CYP19A1 (0.35)
SCHEMBL11046890 0.79 CYP19A1 (0.36) MEN1KMT2ATSHRMAPK1
SCHEMBL11057231 0.77
SCHEMBL11042162 0.77 TOP2A (0.34) LMNASMN1; SMN2ALDH1A1
SCHEMBL11045300 0.77 P2RX7 (0.33)
SCHEMBL11044703 0.76 AR (0.31)
SCHEMBL11043196 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0122452-A1 Triazolyl- and imidazolyl-substituted fluoroalkane derivatives, process for their preparation and pharmaceutical compositions containing them SCHERING CORPORATION (US) 1984-10-24 EP disclosed