SCHEMBL11044384

SCHEMBL11044384

Cc1ccc(NC(=O)ONC2=Nc3ccc(Cl)cc3C(c3ccccc3F)=NC2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.41
LMNA P02545 1/20 0.40
THRB P10828 1/20 0.40
DRD3 P35462 2/20 0.39
OPRK1 P41145 2/20 0.39
SLC22A1 O15245 1/20 0.39
ABCB11 O95342 1/20 0.39
CYP3A4 P08684 1/20 0.39
PDE4D Q08499 1/20 0.39
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
AURKA O14965 1/20 0.38
CHRM1 P11229 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTR1A P08908 1/20 0.36
HTR3A P46098 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11169123 0.92 LMNA (0.42) TP53LMNACYP3A4AURKACHRM1
SCHEMBL11039376 0.90 TP53 (0.46) TP53LMNACYP3A4MEN1KMT2A
SCHEMBL11053089 0.90 LMNA (0.44) TP53LMNADRD3OPRK1SLC22A1
SCHEMBL11057804 0.89 LMNA (0.44) TP53LMNADRD3OPRK1SLC22A1
SCHEMBL11160221 0.88 TP53 (0.44) TP53LMNACYP3A4MEN1KMT2A
SCHEMBL11162886 0.88 LMNA (0.43) TP53LMNADRD3OPRK1SLC22A1
SCHEMBL11046042 0.86 TP53 (0.43) TP53LMNAMEN1KMT2AAURKA
SCHEMBL11169424 0.85 GABRA1 (0.40) TP53LMNAMEN1KMT2AAURKA
SCHEMBL11041566 0.84 GABRA1 (0.41) TP53LMNACYP3A4GAAKMT2A
SCHEMBL11168051 0.84 GABRA1 (0.41) TP53LMNAOPRK1PDE4DMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0041242-B1 CARBAMOYLOXYAMINO-1,4-BENZODIAZEPINES, THEIR PREPARATION AND MEDICINES CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1984-07-11 EP disclosed
US-4395409-A ANXIOLYTIC AGENT HOECHST AKTIENGESELLSCHAFT (DE) 1983-07-26 US disclosed