SCHEMBL11044558

SCHEMBL11044558

Cc1c(C(=O)c2ccccc2)[nH]c(Br)c1Br.O=C(c1ccccc1)c1cc(Br)c(Br)[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.40
CYP1A2 P05177 2/20 0.39
HPGD P15428 2/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC10 Q969S8 2/20 0.36
HDAC11 Q96DB2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11003325 0.84 MAP2K1 (0.53) MAP2K1CYP1A2HPGDCYP2D6CYP2C19
SCHEMBL11006723 0.75 ALDH1A1 (0.50) HPGDMEN1KMT2AHDAC6RAB9A
SCHEMBL11052447 0.73 LTA4H (0.40) CYP1A2HPGDMEN1KMT2ACYP3A4
SCHEMBL10939267 0.70 ALDH1A1 (0.45) CYP1A2HPGDCYP2D6CYP2C19MEN1
SCHEMBL11867579 0.69 MEN1 (0.56) MAP2K1CYP1A2HPGDMEN1KMT2A
SCHEMBL11868641 0.69 MEN1 (0.56) CYP1A2MEN1KMT2AHDAC6CYP3A4
SCHEMBL11008783 0.68 L3MBTL1 (0.40) HPGDALDH1A1L3MBTL1
SCHEMBL15197094 0.66 MEN1 (0.46) CYP1A2HPGDMEN1KMT2AHDAC6
SCHEMBL2915910 0.66 GPR35 (0.46) CYP1A2HPGDCYP2C19MEN1KMT2A
SCHEMBL1518075 0.64 MAP2K1 (0.65) MAP2K1HPGDCYP2C19MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4456759-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIPYRETICS, ANTICOAGULANTS, AND MUSCLE RELAXANTS SYNTEX (U.S.A.) INC. (US) 1984-06-26 US disclosed
US-4347185-A DECARBOXYLATION OF THE 1,1-DICARBOXYLATES SYNTEX (U.S.A.) INC. (US) 1982-08-31 US disclosed