SCHEMBL11045005

SCHEMBL11045005

COc1ccc2c(c1)CCN2Cc1cccc(CN)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
NOTUM Q6P988 1/20 0.44
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
PRMT6 Q96LA8 1/20 0.43
MAOB P27338 2/20 0.43
SIGMAR1 Q99720 1/20 0.43
PTGER4 P35408 1/20 0.42
PTGER2 P43116 1/20 0.42
ADRB2 P07550 2/20 0.42
ADRB1 P08588 2/20 0.42
ADRB3 P13945 2/20 0.42
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
ALDH1A1 P00352 2/20 0.42
GAA P10253 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10636985 0.99 HDAC1 (0.47) HDAC1HDAC6NOTUMITGB3ITGA2B
SCHEMBL8815909 0.85 HDAC1 (0.56) HDAC1HDAC6NOTUMSIGMAR1ADRB2
SCHEMBL10636799 0.83 SCN5A (0.50) HDAC1HDAC6NOTUMMAOBSIGMAR1
SCHEMBL11041268 0.81 HSD17B3 (0.47) HDAC1HDAC6NOTUMPRMT6SIGMAR1
SCHEMBL11041562 0.80 SRD5A1 (0.45) NOTUMMAOBADRB2ADRB1ADRB3
SCHEMBL11013870 0.80 ALDH1A1 (0.53) HDAC1HDAC6PRMT6ALDH1A1GAA
SCHEMBL5661589 0.79 SIGMAR1 (0.57) SIGMAR1PTGER4PTGER2ALDH1A1GAA
SCHEMBL12628333 0.79 HDAC1 (0.58) HDAC1HDAC6NOTUMADRB2ADRB1
SCHEMBL29572755 0.79 SIGMAR1 (0.57) SIGMAR1PTGER4PTGER2ALDH1A1GAA
Hydrochloric Acid SCHEMBL10642538 0.79 EGFR (0.46) NOTUMMAOBADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4448784-A 1-(Aminoalkylphenyl and aminoalkylbenzyl)-indoles and indolines and analgesic method of use thereof HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1984-05-15 US claimed