SCHEMBL11045896

SCHEMBL11045896

CSc1nc(-c2ccccc2)c(-c2ccccc2)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.55
MAPT P10636 4/20 0.55
CYP1A2 P05177 2/20 0.55
CYP2D6 P10635 2/20 0.55
CYP2C19 P33261 2/20 0.55
HRH3 Q9Y5N1 1/20 0.49
KDM4E B2RXH2 2/20 0.49
CYP3A4 P08684 1/20 0.49
GAA P10253 1/20 0.49
CYP2C9 P11712 1/20 0.49
NPSR1 Q6W5P4 3/20 0.44
PTGS2 P35354 4/20 0.44
PTGS1 P23219 2/20 0.44
KMT2A Q03164 4/20 0.43
LMNA P02545 3/20 0.43
MEN1 O00255 3/20 0.43
MAPK1 P28482 2/20 0.43
XIAP P98170 1/20 0.42
HPGD P15428 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11038402 0.86 ALOX5 (0.44) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL7621307 0.86 ALOX5 (0.48) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL11040057 0.82 PTGS2 (0.48) ALDH1A1MAPTKDM4EGAANPSR1
SCHEMBL11707308 0.81 ALDH1A1 (0.51) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL11704670 0.81 HTR7 (0.60) ALDH1A1MAPTCYP1A2CYP2C19CYP2C9
SCHEMBL11040051 0.81 ALDH1A1 (0.58) ALDH1A1MAPTCYP1A2KDM4ECYP3A4
SCHEMBL11040891 0.81 HRH3 (0.56) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL10787518 0.80 PTGS1 (0.52) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL543986 0.80 ALDH1A1 (0.44) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL11039848 0.80 HRH3 (0.58) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0061425-A2 Thiazole derivatives, processes for their preparation, medicaments containing them and their use CIBA-GEIGY AG (CH) 1982-09-29 EP claimed
US-4451471-A Certain 2,4,5-tri-substituted thiazoles, pharmaceutical compositions containing same and methods of using same CIBA-GEIGY CORPORATION (US) 1984-05-29 US disclosed
EP-0061425-A2 Thiazole derivatives, processes for their preparation, medicaments containing them and their use CIBA-GEIGY AG (CH) 1982-09-29 EP disclosed
US-4022607-A Substituted oxazoles and thiazoles as herbicides SANDOZ, INC. (US) 1977-05-10 US disclosed