SCHEMBL11048397

SCHEMBL11048397

COc1ccc(-c2c[nH]c(CO)n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.47
NPC1 O15118 8/20 0.45
RAB9A P51151 7/20 0.45
MAPK1 P28482 2/20 0.43
MAPT P10636 7/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
ALDH1A1 P00352 4/20 0.42
POLB P06746 3/20 0.42
FYN P06241 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 4/20 0.41
LMNA P02545 2/20 0.41
PKM P14618 2/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
DYRK1A Q13627 1/20 0.41
CASP3 P42574 1/20 0.41
SENP7 Q9BQF6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10886759 0.85 PDGFRB (0.46) PDGFRBNPC1RAB9AMAPK1MAPT
SCHEMBL10099697 0.84 PDGFRB (0.50) PDGFRBNPC1RAB9AMAPTSMN1; SMN2
SCHEMBL11047835 0.83 METAP2 (0.38) NPC1RAB9AMAPTSMN1; SMN2ALDH1A1
SCHEMBL11048359 0.80 METAP2 (0.44) PDGFRBNPC1RAB9AMAPTSMN1; SMN2
SCHEMBL7487071 0.80 ADORA3 (0.41) MAPTALDH1A1KDM4E
SCHEMBL15818572 0.79 MAPK1 (0.38) NPC1RAB9AMAPK1SMN1; SMN2ALDH1A1
SCHEMBL855275 0.79 METAP2 (0.38) NPC1RAB9AMAPTSMN1; SMN2ALDH1A1
SCHEMBL11049905 0.79 NOTUM (0.47) PDGFRBMAPTALDH1A1MEN1KMT2A
SCHEMBL8656607 0.79 MAOB (0.43) PDGFRBNPC1RAB9AMAPK1MAPT
SCHEMBL4878975 0.79 NOTUM (0.44) PDGFRBRAB9AMAPK1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024829-B1 4-BENZYL- AND 4-BENZOYLIMIDAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Farmos-Yhtyma Oy (FI) 1984-04-25 EP claimed
US-4443466-A DIURETICS, SEDATIVES, ANALGESICS Farmos-Yhtyma OY (Farmos Group Ltd.) (FI) 1984-04-17 US claimed
EP-0024829-A1 4-Benzyl- and 4-benzoylimidazole derivatives, processes for their preparation and pharmaceutical compositions comprising the same Farmos-Yhtyma Oy (FI) 1981-03-11 EP claimed
EP-0024829-B1 4-BENZYL- AND 4-BENZOYLIMIDAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Farmos-Yhtyma Oy (FI) 1984-04-25 EP disclosed
US-4443466-A DIURETICS, SEDATIVES, ANALGESICS Farmos-Yhtyma OY (Farmos Group Ltd.) (FI) 1984-04-17 US disclosed
EP-0024829-A1 4-Benzyl- and 4-benzoylimidazole derivatives, processes for their preparation and pharmaceutical compositions comprising the same Farmos-Yhtyma Oy (FI) 1981-03-11 EP disclosed