SCHEMBL11052138

SCHEMBL11052138

CC(C)(C)NC(=O)NC(=N)Nc1c(F)cccc1Br

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
LMNA P02545 1/20 0.39
HTT P42858 2/20 0.39
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ANO1 Q5XXA6 2/20 0.36
PDGFRB P09619 2/20 0.35
FGFR1 P11362 2/20 0.35
SRC P12931 2/20 0.35
PDGFRA P16234 2/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11054793 0.92 NPC1 (0.44) KMT2AMEN1NPC1RAB9ALMNA
SCHEMBL11050055 0.90 KMT2A (0.45) KMT2AMEN1NPC1RAB9ALMNA
SCHEMBL11578638 0.86 KMT2A (0.40) KMT2AMEN1NPC1RAB9ALMNA
SCHEMBL11578817 0.86 SMN1; SMN2 (0.39) KMT2AMEN1NPC1RAB9ALMNA
SCHEMBL11056090 0.85 NPC1 (0.39) KMT2AMEN1NPC1RAB9ALMNA
SCHEMBL11056782 0.85 MAPK1 (0.48) KMT2AMEN1NPC1RAB9ALMNA
SCHEMBL11054677 0.85 LMNA (0.40) KMT2AMEN1LMNAHTTMAPK1
SCHEMBL11049616 0.84 HTT (0.50) KMT2AMEN1RAB9ALMNAHTT
SCHEMBL11579645 0.83 PTGS2 (0.41) KMT2AMEN1LMNAHTTMAPK1
SCHEMBL11580574 0.82 TBXA2R (0.39) KMT2AMEN1NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed