SCHEMBL11053014

SCHEMBL11053014

Cc1cccc(Br)c1N(C(=N)N)C(=O)NCCOCCc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HPGD P15428 3/20 0.34
P2RX7 Q99572 1/20 0.34
NLRP3 Q96P20 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
F10 P00742 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
ACHE P22303 2/20 0.32
OPRM1 P35372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11558027 0.92 SMN1; SMN2 (0.39) SMN1; SMN2LMNAL3MBTL1HPGDP2RX7
SCHEMBL11053515 0.91 SMN1; SMN2 (0.41) SMN1; SMN2LMNAL3MBTL1HPGDP2RX7
SCHEMBL11056622 0.88 OPRM1 (0.38) SMN1; SMN2LMNAL3MBTL1HPGDP2RX7
SCHEMBL11057720 0.88 ALDH1A1 (0.39) SMN1; SMN2LMNAL3MBTL1HPGDP2RX7
SCHEMBL11055968 0.85 SMN1; SMN2 (0.39) SMN1; SMN2LMNACYP3A4F10HTT
SCHEMBL11056521 0.84 HPGD (0.40) SMN1; SMN2L3MBTL1HPGDCYP2C9HTT
Hydrochloric Acid SCHEMBL11557076 0.82 SMN1; SMN2 (0.44) SMN1; SMN2LMNAL3MBTL1P2RX7KMT2A
Hydrochloric Acid SCHEMBL11562331 0.81 SMN1; SMN2 (0.44) SMN1; SMN2LMNAHPGDP2RX7HTT
SCHEMBL11057304 0.81 L3MBTL1 (0.38) LMNAL3MBTL1HPGDCYP3A4F10
Hydrochloric Acid SCHEMBL11581693 0.80 ALDH1A1 (0.40) SMN1; SMN2L3MBTL1HPGDCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed