SCHEMBL11053334

SCHEMBL11053334

Cc1cccc(Cl)c1N(C(=N)N)C(=O)NC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HPGD P15428 1/20 0.37
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
ESR1 P03372 2/20 0.36
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
CXCL8 P10145 1/20 0.34
MAPT P10636 2/20 0.33
POLB P06746 2/20 0.33
S1PR4 O95977 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33
SRC P12931 1/20 0.33
MAPK14 Q16539 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11557239 0.89 PKM (0.34) MAPK1MEN1KMT2AALDH1A1MAPT
SCHEMBL10613005 0.86 ESR1 (0.37) KMT2APDK1PDK2PDK3PDK4
Hydrochloric Acid SCHEMBL11053035 0.85 ESR1 (0.36) KMT2APDK1PDK2PDK3PDK4
SCHEMBL11051496 0.84 CA1 (0.32) MEN1KMT2AALDH1A1HTTSRC
SCHEMBL11053340 0.83 ALDH1A1 (0.36) HPGDESR1ALDH1A1CXCL8MAPT
Hydrochloric Acid SCHEMBL11077419 0.83 S1PR4 (0.35) MEN1KMT2AESR1ALDH1A1HTT
SCHEMBL11054047 0.83 ALDH1A1 (0.40) MEN1KMT2AHPGDESR1ALDH1A1
SCHEMBL11059255 0.83 ABL1 (0.40) ESR1ALDH1A1HTTMAPTS1PR4
Hydrochloric Acid SCHEMBL11133882 0.82 ABL1 (0.40) ESR1ALDH1A1HTTMAPTS1PR4
SCHEMBL11053218 0.81 RORC (0.35) KMT2AESR1ALDH1A1MAPTS1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed