SCHEMBL11054561

SCHEMBL11054561

CC(C)(C)NC(=O)NC(=N)Nc1ccc(F)cc1F

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.50
RAB9A P51151 8/20 0.48
NPC1 O15118 7/20 0.48
PKM P14618 3/20 0.48
SMN1; SMN2 Q16637 5/20 0.48
GAA P10253 3/20 0.46
RECQL P46063 1/20 0.46
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
ALDH1A1 P00352 1/20 0.44
CYP2C19 P33261 1/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 2/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11053888 0.89 HTT (0.47) HTTRAB9ANPC1PKMSMN1; SMN2
SCHEMBL11052569 0.87 ALDH1A1 (0.43) HTTRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL11053439 0.87 HTT (0.42) HTTRAB9ANPC1SMN1; SMN2GAA
SCHEMBL11250897 0.86 PKM (0.48) HTTRAB9ANPC1PKMSMN1; SMN2
SCHEMBL11053772 0.86 HTT (0.38) HTTRAB9ANPC1PKMSMN1; SMN2
SCHEMBL11052091 0.86 NPC1 (0.40) HTTRAB9ANPC1PKMSMN1; SMN2
SCHEMBL11052904 0.86 HTT (0.47) HTTPOLB
SCHEMBL11049781 0.86 KIF11 (0.46) HTTSMN1; SMN2LMNA
SCHEMBL11053656 0.86 HTT (0.50) HTTRAB9ANPC1PKMSMN1; SMN2
SCHEMBL11055911 0.86 HTT (0.41) HTTRAB9ANPC1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed