SCHEMBL11050195

SCHEMBL11050195

CNc1ncn(-c2c(C)cccc2C)c(=S)n1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.39
CHRNA7 P36544 9/20 0.33
CXCR2 P25025 1/20 0.31
EGFR P00533 1/20 0.30
FGFR1 P11362 1/20 0.30
SRC P12931 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11057092 0.90 CHRNA7 (0.44) HCAR1CHRNA7EGFRFGFR1SRC
SCHEMBL11054223 0.88 KMT2A (0.36) HCAR1CHRNA7
SCHEMBL11058209 0.85 HCAR1 (0.38) HCAR1CHRNA7SRC
SCHEMBL11059281 0.84 KDM4E (0.37)
SCHEMBL11053099 0.84 HCAR1 (0.37) HCAR1CHRNA7FGFR1
SCHEMBL11054647 0.84 HCAR1 (0.37) HCAR1CHRNA7EGFRFGFR1
SCHEMBL11061839 0.84 HCAR1 (0.37) HCAR1CHRNA7
SCHEMBL11061669 0.82 WEE1 (0.44) CHRNA7FGFR1SRC
SCHEMBL11053291 0.81 HCAR1 (0.35) HCAR1CHRNA7EGFRFGFR1
SCHEMBL11054404 0.81 HCAR1 (0.46) HCAR1CHRNA7EGFRFGFR1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed