SCHEMBL11056407

SCHEMBL11056407

CNc1ncn(-c2c(C)cc(C)cc2C)c(=O)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.34
HCAR1 Q9BXC0 3/20 0.31
CHRNA7 P36544 1/20 0.31
TP53 P04637 2/20 0.30
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
KDM4A O75164 1/20 0.30
ALDH1A1 P00352 1/20 0.30
ABL1 P00519 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
CDH1 P12830 1/20 0.30
TCF4 P15884 1/20 0.30
TSHR P16473 1/20 0.30
APC P25054 1/20 0.30
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11060337 0.90 CRHR1 (0.33) CRHR1
SCHEMBL11050289 0.88 ESR1 (0.39)
SCHEMBL11055502 0.88 AURKA (0.32)
SCHEMBL11050393 0.87 ESR1 (0.31) CRHR1KDM4ENPC1ALDH1A1RAB9A
SCHEMBL11474313 0.85 MEN1 (0.31) NPC1LMNARAB9AKMT2ANOS3
SCHEMBL11054404 0.84 HCAR1 (0.46) HCAR1CHRNA7ALDH1A1POLBKMT2A
SCHEMBL11351070 0.84 ALDH1A1 (0.41) CRHR1TP53KDM4EALDH1A1LMNA
Hydrochloric Acid SCHEMBL11052665 0.83 HCAR1 (0.44) HCAR1CHRNA7ALDH1A1POLBKMT2A
SCHEMBL11059281 0.81 KDM4E (0.37) CRHR1KDM4EALDH1A1NOS3NOS2
SCHEMBL11058230 0.79 ESR1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed