SCHEMBL11056546

SCHEMBL11056546

Cc1cc(C(F)(F)F)cc(Cl)c1NC(=O)NC(=N)N

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 1/20 0.38
MAPT P10636 2/20 0.37
ALDH1A1 P00352 4/20 0.37
RXFP1 Q9HBX9 1/20 0.37
GAA P10253 2/20 0.36
GPR35 Q9HC97 3/20 0.36
KMT2A Q03164 2/20 0.36
RAPGEF4 Q8WZA2 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11140619 0.84 ALDH1A1 (0.42) HTTL3MBTL1MAPTALDH1A1GAA
SCHEMBL11278607 0.83 HTT (0.39) HTTL3MBTL1TSHRMAPTALDH1A1
SCHEMBL11286642 0.83 HTT (0.55) HTTL3MBTL1TSHRMAPTALDH1A1
SCHEMBL11059296 0.83 RAPGEF4 (0.42) HTTL3MBTL1TSHRMAPTALDH1A1
Hydrochloric Acid SCHEMBL11414461 0.82 RAPGEF4 (0.41) HTTL3MBTL1TSHRMAPTALDH1A1
SCHEMBL10732669 0.82 HTT (0.40) HTTL3MBTL1TSHRMAPTALDH1A1
SCHEMBL11428458 0.81 HTT (0.40) HTTL3MBTL1TSHRMAPTALDH1A1
SCHEMBL11279723 0.81 HTT (0.42) HTTL3MBTL1TSHRMAPTALDH1A1
SCHEMBL11052671 0.80 KDR (0.38) HTTMAPTGAARAPGEF4LMNA
SCHEMBL11274752 0.80 TSHR (0.44) HTTL3MBTL1TSHRMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed