SCHEMBL11279723

SCHEMBL11279723

Cc1cc(Br)cc(Cl)c1NC(=O)NC(=N)N

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 6/20 0.41
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.40
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HPGD P15428 2/20 0.39
POLB P06746 1/20 0.39
IDH1 O75874 1/20 0.39
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
DRD2 P14416 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2B P41595 1/20 0.36
PKM P14618 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11192133 0.90 CYP1A2 (0.36) HTTTSHRMAPTKMT2ALMNA
SCHEMBL11055179 0.90 ALDH1A1 (0.48) ALDH1A1MAPTKMT2ALMNAHPGD
SCHEMBL11280868 0.89 IDH1 (0.38) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL11286642 0.88 HTT (0.55) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL11282636 0.85 HTT (0.38) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL11434842 0.85 CYP1A2 (0.33) HTTALDH1A1MAPTKMT2ALMNA
SCHEMBL11059296 0.85 RAPGEF4 (0.42) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL10854903 0.85 HTT (0.41) HTTTSHRALDH1A1MAPTKMT2A
SCHEMBL11052411 0.84 HTT (0.41) HTTTSHRALDH1A1MAPTKMT2A
Hydrochloric Acid SCHEMBL11414461 0.84 RAPGEF4 (0.41) HTTTSHRALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4283555-A Amidinoureas WILLIAM H. RORER, INC. (US) 1981-08-11 US disclosed
US-4216229-A 1-AMIDINO-3-PHENYLUREAS WILLIAM H. RORER, INC. (US) 1980-08-05 US disclosed
US-4216230-A Method for alleviating hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-08-05 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4183956-A Method for treating gastrointestinal spasms, gastrointestinal hyperacidity and hypertensive disorders with amidinoureas WILLIAM H. RORER, INC. (US) 1980-01-15 US disclosed
US-4150154-A GASTROINTESTINAL ANTISPASMODICS WILLIAM H. RORER, INC. (US) 1979-04-17 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed