SCHEMBL11060055

SCHEMBL11060055

Cc1ccc(C2CC(N)=NN2c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.53
ERBB2 P04626 2/20 0.53
ERBB3 P21860 1/20 0.53
KDR P35968 1/20 0.53
PTK2 Q05397 1/20 0.53
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
PRKCZ Q05513 2/20 0.49
MAOA P21397 4/20 0.49
MAOB P27338 4/20 0.49
PDE5A O76074 1/20 0.47
MAPT P10636 4/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 2/20 0.46
LMNA P02545 1/20 0.46
ATM Q13315 2/20 0.44
HSP90AA1 P07900 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11068412 0.89 MEN1 (0.54) EGFRERBB2CA1CA2PRKCZ
SCHEMBL11060811 0.84 PRKCZ (0.56) EGFRERBB2CA1CA2PRKCZ
SCHEMBL11374953 0.84 PRKCZ (0.53) EGFRERBB2ERBB3KDRPTK2
SCHEMBL8637990 0.84 PRKCZ (0.46) EGFRERBB2ERBB3KDRPTK2
SCHEMBL10418603 0.84 PRKCZ (0.46) EGFRERBB2PRKCZMAPTMEN1
SCHEMBL25138590 0.80 EGFR (0.78) EGFRERBB2ERBB3KDRPTK2
SCHEMBL11096598 0.79 EGFR (0.48) EGFRERBB2ERBB3KDRPTK2
SCHEMBL908494 0.78 CA1 (0.56) EGFRERBB2CA1CA2PRKCZ
SCHEMBL11064115 0.78 MEN1 (0.58) EGFRERBB2CA1CA2PRKCZ
SCHEMBL11101684 0.78 ALDH1A1 (0.65) EGFRERBB2CA1CA2PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447442-A ANTIINFLAMMATORY, ANTIARTHRITIC, ANTIHISTAMINE, ANTIALLERGENS, ANALGESICS, BACTERICIDES, AND FUNGICIDES AMERICAN CYANAMID COMPANY (US) 1984-05-08 US disclosed
US-4432991-A ANALGESICS, FUNGICIDE, BACTERICIDE, ANTIINFLAMMATORY, OR ANTIARTHRITIC AGENTS, ANTIALLERGENS, AND BRONCHODILATOR AMERICAN CYANAMID COMPANY (US) 1984-02-21 US disclosed
EP-0070376-A1 Heterocyclic substituted-amino-pyrazolines AMERICAN CYANAMID COMPANY (US) 1983-01-26 EP disclosed
US-4360680-A ANALGESIC, ANTIINFLAMMATORY AGENT, FUNGICIDE AND BACTERICIDE AMERICAN CYANAMID COMPANY (US) 1982-11-23 US disclosed
US-4348527-A ANALGESICS, BACTERICIDES, FUNGICIDES AMERICAN CYANAMID COMPANY (US) 1982-09-07 US disclosed