SCHEMBL11060091

SCHEMBL11060091

CCCNC(=O)N(C(=N)N)c1c(C)cccc1CC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
TP53 P04637 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
CYP3A4 P08684 1/20 0.41
ESR1 P03372 1/20 0.36
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34
GABRA2 P47869 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
EPHX1 P07099 1/20 0.34
NR1I2 O75469 1/20 0.34
PTGES O14684 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
MTNR1A P48039 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11054316 0.95 TP53 (0.37) ALDH1A1TP53TDP1CYP3A4MEN1
SCHEMBL11056672 0.93 POLB (0.41) ALDH1A1TP53TDP1CYP3A4ESR1
SCHEMBL11057738 0.91 TDP1 (0.39) ALDH1A1TP53TDP1CYP3A4MEN1
Hydrochloric Acid SCHEMBL11565511 0.91 GABRG2 (0.36) ALDH1A1TP53TDP1CYP3A4GABRG2
SCHEMBL11056380 0.90 ALDH1A1 (0.40) ALDH1A1TP53TDP1CYP3A4ESR1
SCHEMBL11096045 0.88 ALDH1A1 (0.41) ALDH1A1TP53TDP1CYP3A4MEN1
SCHEMBL11053069 0.87 POLB (0.45) ALDH1A1TP53TDP1MEN1KMT2A
SCHEMBL11060262 0.86 NR1I2 (0.38) ALDH1A1TP53TDP1CYP3A4MEN1
SCHEMBL11057304 0.86 L3MBTL1 (0.38) ALDH1A1TP53TDP1CYP3A4KMT2A
SCHEMBL11054409 0.86 ESR1 (0.39) ALDH1A1TP53TDP1CYP3A4ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed