SCHEMBL11060185

SCHEMBL11060185

CCc1cccc(CC)c1-n1cnc(N(CC)OCc2ccccc2)nc1=S

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
C5AR1 P21730 1/20 0.33
BCHE P06276 4/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CRHR1 P34998 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
GAA P10253 1/20 0.31
STAT3 P40763 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056353 0.89 HCAR2 (0.34) ALDH1A1MEN1KMT2ACRHR1HCAR2
SCHEMBL11055462 0.89 HCAR2 (0.35) ALDH1A1C5AR1BCHECRHR1HCAR2
SCHEMBL11059465 0.83 KMT2A (0.37) MEN1KMT2ACRHR1HCAR2MAOA
SCHEMBL11053513 0.82 MAPK14 (0.39) ALDH1A1MEN1KMT2AHCAR2HPGD
SCHEMBL11056509 0.81 GRM1 (0.34) ALDH1A1KMT2AESR1ESR2LMNA
SCHEMBL11059482 0.78 HCAR2 (0.37) ALDH1A1KMT2ACRHR1HCAR2LMNA
SCHEMBL11057683 0.74 MAPK14 (0.34) MEN1KMT2ASTAT3HTTSMN1; SMN2
SCHEMBL11059306 0.74 CHRNA7 (0.45) ALDH1A1HPGDMAPK14
SCHEMBL11060192 0.73 MKNK1 (0.36) ALDH1A1MEN1KMT2ACRHR1HTT
SCHEMBL11056312 0.73 LCK (0.44) ALDH1A1MEN1KMT2ALMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed