SCHEMBL11059306

SCHEMBL11059306

CCN(OCc1ccccc1)c1ncn(-c2c(C)cccc2Cl)c(=O)n1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 11/20 0.45
MAPK14 Q16539 2/20 0.40
P2RX7 Q99572 1/20 0.36
FABP3 P05413 1/20 0.36
FABP4 P15090 1/20 0.36
FABP5 Q01469 1/20 0.36
LCK P06239 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11053513 0.91 MAPK14 (0.39) CHRNA7MAPK14P2RX7FABP3FABP4
SCHEMBL11055027 0.90 CHRNA7 (0.44) CHRNA7MAPK14P2RX7KDM4EALDH1A1
SCHEMBL11056305 0.90 MEN1 (0.38) CHRNA7MAPK14P2RX7
SCHEMBL11057683 0.88 MAPK14 (0.34) CHRNA7MAPK14P2RX7
SCHEMBL11055462 0.85 HCAR2 (0.35) MAPK14ALDH1A1HPGD
SCHEMBL11055569 0.80 CHRNA7 (0.43) CHRNA7LCK
SCHEMBL11059411 0.80 KMT2A (0.36) CHRNA7ALDH1A1
SCHEMBL11052478 0.78 TDP2 (0.33) CHRNA7MAPK14P2RX7ALDH1A1HPGD
SCHEMBL11060185 0.74 ALDH1A1 (0.33) MAPK14ALDH1A1HPGD
SCHEMBL11059482 0.74 HCAR2 (0.37) P2RX7ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed