SCHEMBL11060269

SCHEMBL11060269

Nc1ncn(-c2ccc(C(F)(F)F)cc2)c(=S)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
DHFR P00374 2/20 0.46
CDC7 O00311 1/20 0.39
CDK2 P24941 1/20 0.39
LCK P06239 1/20 0.39
KIT P10721 1/20 0.39
SRC P12931 1/20 0.39
KDR P35968 1/20 0.39
CYP11B2 P19099 1/20 0.38
XDH P47989 2/20 0.38
HSP90B1 P14625 1/20 0.36
TRAP1 Q12931 1/20 0.36
PI4KA P42356 1/20 0.35
PI4K2B Q8TCG2 1/20 0.35
PI4K2A Q9BTU6 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
KIF11 P52732 1/20 0.35
GFER P55789 1/20 0.35
NOTUM Q6P988 1/20 0.35
JAK2 O60674 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18284894 0.71 DHFR (0.42) TDP1DHFRSRCKDRXDH
SCHEMBL31013386 0.70 NOTUM (0.43) TDP1DHFRSRCKDRXDH
SCHEMBL11058394 0.69 PI4KA (0.34) TDP1PI4KAPI4K2BPI4K2API4KB
SCHEMBL8845189 0.66 TDP1 (0.45) TDP1DHFRCDK2SRCKDR
SCHEMBL6603766 0.66 ALOX15B (0.46) TDP1DHFRCYP11B2XDHKIF11
SCHEMBL28281841 0.65 DHFR (0.49) DHFRCDC7CDK2LCKKIT
SCHEMBL11060314 0.65 PI4KA (0.49) TDP1PI4KAPI4K2BPI4K2API4KB
SCHEMBL28848076 0.65 JAK2 (0.43) TDP1DHFRCDK2SRCKDR
SCHEMBL30723122 0.63 HTT (0.68) KDRCYP1A2CYP2C19KDM4EALDH1A1
SCHEMBL29145142 0.63 HTT (0.68) KDRCYP1A2CYP2C19KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed