SCHEMBL8845189

SCHEMBL8845189

Nc1nncn1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
KIF11 P52732 2/20 0.39
NOTUM Q6P988 1/20 0.38
XDH P47989 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
DHFR P00374 1/20 0.37
NOD1 Q9Y239 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP11B2 P19099 1/20 0.35
SRC P12931 1/20 0.35
BRAF P15056 1/20 0.35
KDR P35968 1/20 0.35
PTGS2 P35354 1/20 0.35
P2RX7 Q99572 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21597614 0.81 NPC1 (0.41) TDP1NOTUMMAPTRAB9ACYP11B2
SCHEMBL2545002 0.78 TDP1 (0.45) TDP1KIF11NOTUMMAPTRAB9A
SCHEMBL14710285 0.77 POLB (0.39) TDP1RAB9A
SCHEMBL544340 0.76 MAPK1 (0.41) NOTUMMAPTEGFR
SCHEMBL8389202 0.70 OPRD1 (0.54) TDP1KIF11RAB9APTGS2
SCHEMBL11595644 0.70 SCN5A (0.43) TDP1KIF11NOTUMCYP11B2
SCHEMBL28452141 0.69 MAPT (0.48) TDP1KIF11NOTUMXDHMKNK1
SCHEMBL11060269 0.66 TDP1 (0.47) TDP1KIF11NOTUMXDHDHFR
SCHEMBL18284894 0.66 DHFR (0.42) TDP1KIF11NOTUMXDHDHFR
SCHEMBL11594125 0.66 MAPK1 (0.40) NOTUMMAPTCYP11B2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5674886-A AROMATASE INHIBITOR; BREAST CANCER; UROGENITAL DISORDERS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-10-07 US disclosed