SCHEMBL11061534

SCHEMBL11061534

CCc1ccc2c(O)c(C(=O)O)cnc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.43
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
GABRB2 P47870 1/20 0.42
GABRA4 P48169 1/20 0.42
GABRE P78334 1/20 0.42
GABRA6 Q16445 1/20 0.42
GABRG1 Q8N1C3 1/20 0.42
GABRG3 Q99928 1/20 0.42
GABRQ Q9UN88 1/20 0.42
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10032038 0.88 TP53 (0.51) TP53GABRPGABRDGABRA1GABRB1
SCHEMBL7758342 0.85 HMGB1 (0.39) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL10341241 0.85 MEN1 (0.46) GABRA1GABRB2ALDH1A1SMN1; SMN2MEN1
SCHEMBL5766222 0.80 ALDH1A1 (0.47) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL31668736 0.80 KDM4E (0.54) TP53ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL27903036 0.80 CA12 (0.44) ALDH1A1MEN1KMT2AHMGB1CXCL12
SCHEMBL10202030 0.79 KDM4E (0.41) ALDH1A1MEN1KMT2ATSHRPOLB
SCHEMBL11707476 0.79 TP53 (0.48) TP53ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL29952565 0.79 AKR1C3 (0.41) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2724263 0.77 HTT (0.45) ALDH1A1MEN1KMT2ARXFP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447435-A HYPOTENSIVE AGENTS THE BOOTS COMPANY PLC (GB) 1984-05-08 US disclosed
US-4442109-A 3-Methylthiomethyl-and 3-methylsulfinylmethyl-4-quinolinones useful for treating hypertension THE BOOTS COMPANY LIMITED (GB) 1984-04-10 US disclosed
US-4442029-A PEPTIDE SYNTHESIS USING AN ISONITRILE AS ACTIVATOR MARQUARDING DIETER (DE) 1984-04-10 US disclosed