SCHEMBL11063136

SCHEMBL11063136

CCc1c2c(n(C)c1CC(=O)O)-c1c(cc(Cl)ccc1=O)CC2

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.34
PTGS2 P35354 3/20 0.34
ALOX5 P09917 3/20 0.34
PTGS1 P23219 3/20 0.34
NOTUM Q6P988 2/20 0.33
SIRT1 Q96EB6 1/20 0.32
ABCB11 O95342 1/20 0.32
SRD5A1 P18405 2/20 0.32
SRD5A2 P31213 2/20 0.32
ABCB1 P08183 1/20 0.31
OXER1 Q8TDS5 1/20 0.31
HSD17B3 P37058 1/20 0.31
WDR5 P61964 1/20 0.31
PTGES O14684 1/20 0.30
ALOX5AP P20292 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11072105 0.87 SRD5A1 (0.35) PTGS2ALOX5PTGS1NOTUMABCB11
SCHEMBL11060030 0.79 LMNA (0.36)
SCHEMBL11066774 0.72 SRD5A1 (0.43) SRD5A1SRD5A2
SCHEMBL11063950 0.71 PTGS2 (0.33) PTGS2ALOX5PTGS1ABCB11OXER1
SCHEMBL11062697 0.69 LMNA (0.40)
SCHEMBL11065609 0.65 HRH1 (0.39) ABCB11SRD5A1SRD5A2ABCB1
SCHEMBL11064537 0.64 AKR1B1 (0.45) PTGS2ABCB11SRD5A1SRD5A2
SCHEMBL8607662 0.61 PTGS2 (0.57) PTGDR2PTGS2PTGS1ABCB11SRD5A2
SCHEMBL11066911 0.61 KDM1A (0.41) ALOX5ABCB11SRD5A1SRD5A2ABCB1
SCHEMBL509958 0.59 PTGDR2 (0.46) PTGDR2PTGS2ABCB11ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4440779-A Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO., INC. (US) 1984-04-03 US disclosed
EP-0068460-A1 Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO. INC. (US) 1983-01-05 EP disclosed