SCHEMBL11060030

SCHEMBL11060030

CCOC(=O)Cc1c(C(=O)O)c2c(n1C)-c1c(cc(Cl)ccc1=O)CC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
ALDH1A1 P00352 4/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
USP2 O75604 1/20 0.34
HTT P42858 1/20 0.34
SLC2A2 P11168 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HRH1 P35367 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11063299 0.92 ALDH1A1 (0.38) LMNAL3MBTL1ALDH1A1CYP1A2CYP3A4
SCHEMBL11072105 0.89 SRD5A1 (0.35) L3MBTL1TDP1
SCHEMBL11065609 0.87 HRH1 (0.39) LMNAL3MBTL1ALDH1A1CYP1A2CYP3A4
SCHEMBL11062697 0.80 LMNA (0.40) LMNAL3MBTL1ALDH1A1CYP1A2CYP3A4
SCHEMBL11066911 0.80 KDM1A (0.41) LMNAL3MBTL1ALDH1A1CYP1A2CYP3A4
SCHEMBL11063136 0.79 PTGDR2 (0.34)
SCHEMBL11068179 0.77 L3MBTL1 (0.45) LMNAL3MBTL1ALDH1A1MAPTMEN1
SCHEMBL11073141 0.77 AKR1B1 (0.42) LMNAL3MBTL1ALDH1A1CYP1A2CYP3A4
SCHEMBL11066774 0.77 SRD5A1 (0.43) HTTHRH1SLC6A15
SCHEMBL11065512 0.76 MAPK14 (0.40) LMNAL3MBTL1ALDH1A1CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4440779-A Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO., INC. (US) 1984-04-03 US disclosed
EP-0068460-A1 Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO. INC. (US) 1983-01-05 EP disclosed