SCHEMBL11071292

SCHEMBL11071292

COc1ccc(C(CC(N)=O)CC(N)=O)cc1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.61
TNF P01375 1/20 0.55
ALDH1A1 P00352 1/20 0.51
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
PARP10 Q53GL7 2/20 0.50
PARP1 P09874 1/20 0.50
PARP2 Q9UGN5 1/20 0.50
PARP4 Q9UKK3 1/20 0.50
FFAR1 O14842 2/20 0.49
ALOX5 P09917 1/20 0.47
AOC3 Q16853 2/20 0.46
FNTA P49354 2/20 0.46
FNTB P49356 2/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12836590 0.91 FFAR1 (0.59) L3MBTL1TNFALDH1A1CA1CA2
SCHEMBL10455508 0.87 L3MBTL1 (0.49) L3MBTL1TNFALDH1A1CA1CA2
SCHEMBL27702953 0.85 TNF (0.55) L3MBTL1TNFCA1CA2PARP10
SCHEMBL28285282 0.85 ALDH1A1 (0.63) L3MBTL1TNFALDH1A1FFAR1
SCHEMBL12883281 0.84 TNF (0.54) L3MBTL1TNFALDH1A1CA1CA2
SCHEMBL3443782 0.84 L3MBTL1 (0.67) L3MBTL1TNFALDH1A1CA1CA2
SCHEMBL2226074 0.83 L3MBTL1 (0.68) L3MBTL1FFAR1FNTAFNTB
SCHEMBL6211904 0.82 L3MBTL1 (0.55) L3MBTL1TNFALDH1A1
SCHEMBL6289377 0.82 TNF (0.52) L3MBTL1TNFCA1CA2PARP10
SCHEMBL4459742 0.82 TNF (0.52) L3MBTL1TNFCA1CA2PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed