SCHEMBL11074658

SCHEMBL11074658

NC(=O)c1cc2c([nH]c1=O)CSCc1cccnc1-2

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.33
PARP1 P09874 2/20 0.33
CSNK1A1 P48729 1/20 0.33
TYRO3 Q06418 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
BTK Q06187 1/20 0.31
KDM4E B2RXH2 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
DRD1 P21728 1/20 0.31
JAK2 O60674 1/20 0.30
RIPK1 Q13546 1/20 0.30
NUDT1 P36639 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7346618 0.85 AURKA (0.36) AURKAPARP1CSNK1A1TYRO3DYRK1B
SCHEMBL7347592 0.76 MAPK14 (0.39) DRD1
SCHEMBL7341393 0.74 KDM4E (0.39) KDM4EDRD1
SCHEMBL7340073 0.72 CSNK1A1 (0.39) PARP1CSNK1A1TYRO3DYRK1BDDB1
SCHEMBL7348959 0.72 CSNK1A1 (0.39) PARP1CSNK1A1TYRO3DYRK1BDDB1
SCHEMBL7339006 0.68 NOTUM (0.44) AURKAPARP1KDM4E
SCHEMBL7340109 0.68 BCAT2 (0.40) AURKAPARP1CSNK1A1TYRO3DYRK1B
SCHEMBL11092286 0.67 AURKB (0.38) AURKATDP1
SCHEMBL10966773 0.67 FBP1 (0.34) CSNK1A1DYRK1BKDM4E
SCHEMBL11067992 0.67 KDM4E (0.41) KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4474786-A CONGESTIVE HEART FAILURE SCHERING CORPORATION (US) 1984-10-02 US disclosed
EP-0102046-A1 Tricyclic lactams, method for making them, pharmaceutical compositions containing them SCHERING CORPORATION (US) 1984-03-07 EP disclosed