SCHEMBL11075658

SCHEMBL11075658

CN(C)Cc1ccc(C=O)s1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
CYP2A6 P11509 3/20 0.40
CYP2C19 P33261 2/20 0.40
CYP2D6 P10635 1/20 0.40
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALOX5 P09917 1/20 0.35
DPP4 P27487 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PARP1 P09874 1/20 0.33
APP P05067 1/20 0.33
CYP2E1 P05181 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2B6 P20813 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008761 0.82 CYP2A6 (0.41) ALDH1A1CYP2A6CYP2C19CYP2D6ALOX5
SCHEMBL25285356 0.80 ALDH1A1 (0.43) ALDH1A1ADRA1DADRA1AADRA1BKDM4E
SCHEMBL158329 0.77
SCHEMBL29020313 0.76 ALDH1A1 (0.44) ALDH1A1CYP2A6CYP2C19ADRA1DADRA1A
SCHEMBL9192828 0.76 ALDH1A1 (0.50) ALDH1A1CYP2A6CYP2C19ADRA1DADRA1A
SCHEMBL11080507 0.75 TBXAS1 (0.53) ALDH1A1CYP2A6CYP2C19CYP2D6ALOX5
SCHEMBL11080502 0.75 TBXAS1 (0.53) ALDH1A1CYP2A6CYP2C19CYP2D6ALOX5
SCHEMBL8701373 0.74 ALDH1A1 (0.38) ALDH1A1CYP2D6ADRA1DADRA1AADRA1B
SCHEMBL1418985 0.73 ALDH1A1 (0.47) ALDH1A1CYP2A6CYP2C19ADRA1DADRA1A
SCHEMBL27982838 0.73 ALDH1A1 (0.47) ALDH1A1CYP2A6CYP2C19ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104640841-B Lipids for therapeutic agent delivery formulations 日东电工株式会社 2018-04-13 CN disclosed
CN-104640841-A Lipids for therapeutic agent delivery formulations NITTO DENKO CORP 2015-05-20 CN disclosed
EP-0039989-B1 PYRIMIDONE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1984-08-29 EP disclosed
US-4388317-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-06-14 US disclosed
EP-0039989-A1 Pyrimidone derivatives, processes for their preparation and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-11-18 EP disclosed