SCHEMBL11076049

SCHEMBL11076049

NC(=O)CC(CC(N)=O)c1cccc(I)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
PKM P14618 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP2C19 P33261 3/20 0.39
THPO P40225 1/20 0.39
RAB9A P51151 1/20 0.39
HIF1A Q16665 1/20 0.39
TNF P01375 1/20 0.38
SLC6A3 Q01959 4/20 0.37
LMNA P02545 2/20 0.37
PMP22 Q01453 1/20 0.37
GABBR2 O75899 1/20 0.37
GABBR1 Q9UBS5 1/20 0.37
F10 P00742 1/20 0.36
DRD3 P35462 2/20 0.35
ADORA3 P0DMS8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11077894 0.79 MEN1 (0.49) ALDH1A1L3MBTL1LMNA
SCHEMBL11087529 0.79 HDAC4 (0.49) ALDH1A1L3MBTL1
SCHEMBL11075538 0.79 PARP1 (0.47) ALDH1A1L3MBTL1CYP1A2CYP2D6SMN1; SMN2
SCHEMBL11079107 0.79 PARP1 (0.47) ALDH1A1L3MBTL1CYP1A2CYP2D6SMN1; SMN2
SCHEMBL11080280 0.77 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2D6SMN1; SMN2PKM
SCHEMBL9105247 0.77 ALDH1A1 (0.63) ALDH1A1L3MBTL1CYP1A2CYP2D6SMN1; SMN2
SCHEMBL11077922 0.76 ALDH1A1 (0.44) ALDH1A1L3MBTL1CYP1A2CYP2D6SMN1; SMN2
SCHEMBL11078438 0.75 IDO1 (0.39) CYP1A2CYP2D6CYP2C19THPORAB9A
SCHEMBL11081195 0.75 PNMT (0.55)
SCHEMBL11082143 0.75 L3MBTL1 (0.75) ALDH1A1L3MBTL1TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed