SCHEMBL11076384

SCHEMBL11076384

N#CCC(CC#N)c1ccccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
NISCH Q9Y2I1 1/20 0.39
ADRB2 P07550 2/20 0.37
ADRB1 P08588 2/20 0.37
AOC3 Q16853 1/20 0.37
TSHR P16473 4/20 0.36
HIF1A Q16665 3/20 0.36
LMNA P02545 2/20 0.36
IDO1 P14902 2/20 0.36
TDO2 P48775 2/20 0.36
IDO2 Q6ZQW0 2/20 0.36
CYP2C19 P33261 2/20 0.36
BLM P54132 2/20 0.36
CYP2C9 P11712 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NR1I2 O75469 1/20 0.36
ABCB11 O95342 1/20 0.36
NR3C1 P04150 1/20 0.36
PGR P06401 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29483408 1.00 ALDH1A1 (0.41) ALDH1A1NISCHADRB2ADRB1AOC3
SCHEMBL10509388 0.89 NISCH (0.46) ALDH1A1NISCHADRB2ADRB1AOC3
SCHEMBL11082537 0.84 PNMT (0.46) ALDH1A1TSHRLMNAIDO1TDO2
SCHEMBL27168749 0.83 ALDH1A1 (0.41) ALDH1A1NISCHADRB2ADRB1AOC3
SCHEMBL28655921 0.82 ALDH1A1 (0.40) ALDH1A1NISCHADRB2ADRB1AOC3
SCHEMBL28996980 0.80 NISCH (0.41) ALDH1A1NISCHADRB2ADRB1AOC3
SCHEMBL17749161 0.80 ADRB2 (0.42) ALDH1A1NISCHADRB2ADRB1AOC3
SCHEMBL18704103 0.80 ADRB2 (0.50) ALDH1A1NISCHADRB2ADRB1AOC3
SCHEMBL11108160 0.78 TP53 (0.39) ALDH1A1TSHRLMNAIDO1CYP3A4
SCHEMBL11076889 0.77 ESR1 (0.35) ALDH1A1TSHRLMNAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112210549-B Nitrilase mutant protein and application thereof in catalytic synthesis of (R) -3-substituted-4-cyanobutyric acid compounds 中国科学院天津工业生物技术研究所 2022-06-10 CN disclosed
CN-112852789-B Nitrilase mutant and application thereof 中国科学院天津工业生物技术研究所 2022-04-05 CN disclosed
CN-111254134-B Nitrile hydrolase mutant and application thereof in (S) -mononitrile monoacid synthesis 中国科学院天津工业生物技术研究所 2021-09-07 CN disclosed
CN-112852789-A Nitrilase mutant and application thereof 中国科学院天津工业生物技术研究所 2021-05-28 CN disclosed
CN-112210549-A Nitrilase mutant protein and application thereof in catalytic synthesis of (R) -3-substituted-4-cyanobutyric acid compounds 中国科学院天津工业生物技术研究所 2021-01-12 CN disclosed
CN-111254134-A Nitrile hydrolase mutant and application thereof in (S) -mononitrile monoacid synthesis 中国科学院天津工业生物技术研究所 2020-06-09 CN disclosed
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed