SCHEMBL11076403

SCHEMBL11076403

C=CCN(CC1CC1)C1(c2ccc(Cl)cc2)CCC(N(CC)c2ccc(Cl)cc2OC)CC1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.35
KCNN4 O15554 1/20 0.33
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
LTC4S Q16873 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11079047 0.91 CRHR1 (0.34) CRHR1
SCHEMBL11071790 0.86 TSHR (0.36) CRHR1ALDH1A1TSHR
SCHEMBL11068867 0.83 CRHR1 (0.34) CRHR1TSHR
SCHEMBL11069371 0.83 TSHR (0.35) CRHR1ALDH1A1TSHR
SCHEMBL11074056 0.80 CRHR1 (0.33) CRHR1TSHR
SCHEMBL11072624 0.80 TSHR (0.35) TSHR
SCHEMBL11072605 0.80 SLC6A4 (0.41) KCNN4
SCHEMBL11078545 0.80 KCNN4 (0.33) CRHR1KCNN4LTC4S
SCHEMBL11071524 0.78 OPRM1 (0.42) TSHR
SCHEMBL11078728 0.77 TSHR (0.35) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447454-A Analgetic compounds, compositions and process of treatment THE UPJOHN COMPANY (US) 1984-05-08 US disclosed
US-4113866-A ANALGETIC COMPOUNDS, COMPOSITIONS AND PROCESS OF TREATMENT THE UPJOHN COMPANY (US) 1978-09-12 US disclosed