SCHEMBL11076879

SCHEMBL11076879

CC(=O)C1CNCCN1c1ccc(Cl)cc1.c1cc2ccc1-2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
ADRB1 P08588 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CNR2 P34972 3/20 0.39
CNR1 P21554 2/20 0.39
CYP2C8 P10632 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTR2C P28335 6/20 0.38
HTR2B P41595 5/20 0.38
MAPKAPK2 P49137 3/20 0.38
SCN5A Q14524 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
HTR2A P28223 4/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27613840 0.83 HTR3E (0.45) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL653537 0.81 MC4R (0.41) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL1012668 0.81 MC4R (0.41) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL7258181 0.80 ADRB1 (0.43) ADRB1
SCHEMBL21382496 0.80 SLC6A2 (0.34) ADRB1HTR2CHTR2BHTR2A
SCHEMBL23244311 0.78 PKM (0.42) MEN1KMT2A
SCHEMBL27744342 0.76 HTR3E (0.41) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL10683759 0.75 ADRB1 (0.56) ADRB1MEN1KMT2A
Trifluoroacetic Acid SCHEMBL1013575 0.74 F2 (0.41) CNR2CNR1CYP2C8CYP2C9CYP2C19
SCHEMBL11983448 0.74 CNR2 (0.55) CNR2CNR1CYP2C8CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4439606-A ANTICHOLESTEROL, ANTILIPEMIC AGENTS AMERICAN CYANAMID COMPANY (US) 1984-03-27 US disclosed
EP-0094498-A2 Antiatherosclerotic 1-piperazine derivatives AMERICAN CYANAMID COMPANY (US) 1983-11-23 EP disclosed