SCHEMBL11077056

SCHEMBL11077056

CCn1c(-c2ccc(N(C)C)c(C)c2)nc2c3ccc(OC)cc3ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK2 Q13002 4/20 0.44
GRIK1 P39086 2/20 0.44
NPSR1 Q6W5P4 3/20 0.42
POLB P06746 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
TSPO P30536 2/20 0.38
DYRK1A Q13627 1/20 0.37
MAPT P10636 4/20 0.37
PTGER4 P35408 4/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
RPS6KA5 O75582 1/20 0.36
TEK Q02763 1/20 0.36
KDM4E B2RXH2 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
ALDH1A1 P00352 2/20 0.34
NPC1 O15118 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11081346 0.86 PARP1 (0.39) GRIK2GRIK1DYRK1AMAPTSMN1; SMN2
SCHEMBL11086321 0.85 GRIK2 (0.52) GRIK2GRIK1NPSR1POLBTDP1
SCHEMBL11497347 0.79 PARP1 (0.38) GRIK2GRIK1TSPODYRK1AMAPT
SCHEMBL11076799 0.75 CASR (0.50) GRIK2GRIK1NPSR1TSPODYRK1A
SCHEMBL11079618 0.74 GRIK2 (0.52) GRIK2GRIK1NPSR1POLBMAPT
SCHEMBL11073152 0.73 HSD17B10 (0.44) TDP1MAPTPTGER4SMN1; SMN2KDM4E
SCHEMBL11290683 0.73 GRIK2 (0.47) GRIK2GRIK1NPSR1POLBTDP1
SCHEMBL11076164 0.72 SHMT2 (0.42) TDP1MAPTKDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL11086416 0.69 PARP1 (0.51) GRIK2GRIK1DYRK1AMAPTSMN1; SMN2
SCHEMBL11081006 0.69 TLR7 (0.40) MAPTPTGER4SMN1; SMN2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4435417-A ANTIINFLAMMATORY AGENTS GRUPPO LEPETIT S.P.A. (IT) 1984-03-06 US disclosed