SCHEMBL11078071

SCHEMBL11078071

COc1cccc(C2(CCC#N)CCCCC2O)c1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 15/20 0.50
SLC6A3 Q01959 7/20 0.50
SLC22A1 O15245 3/20 0.49
SLC6A2 P23975 8/20 0.47
OPRM1 P35372 3/20 0.47
KMT2A Q03164 2/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
MEN1 O00255 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11078094 0.88 SLC6A4 (0.52) SLC6A4SLC6A3SLC22A1SLC6A2OPRM1
SCHEMBL11550699 0.81 SLC22A1 (0.43) SLC6A4SLC22A1SLC6A2OPRM1KMT2A
SCHEMBL7531306 0.80 SLC6A4 (0.73) SLC6A4SLC6A3SLC22A1SLC6A2OPRM1
SCHEMBL11081655 0.76 SLC6A4 (0.48) SLC6A4SLC6A3SLC22A1SLC6A2OPRM1
SCHEMBL7548669 0.73 SLC6A3 (0.67) SLC6A4SLC6A3SLC6A2
SCHEMBL6851762 0.70 SLC6A4 (0.60) SLC6A4SLC6A3SLC22A1SLC6A2OPRM1
SCHEMBL6851754 0.70 SLC6A4 (0.60) SLC6A4SLC6A3SLC22A1SLC6A2OPRM1
SCHEMBL6851749 0.70 SLC6A4 (0.60) SLC6A4SLC6A3SLC22A1SLC6A2OPRM1
SCHEMBL6851765 0.70 SLC6A4 (0.60) SLC6A4SLC6A3SLC22A1SLC6A2OPRM1
SCHEMBL11079591 0.70 KMT2A (0.43) SLC6A4SLC6A3SLC22A1SLC6A2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4448991-A ANALGESICS HOFFMANN-LA ROCHE INC. (US) 1984-05-15 US disclosed
US-4336268-A Cyclohexene derivative analgesics HOFFMANN-LA ROCHE INC. (US) 1982-06-22 US disclosed
EP-0033156-A2 1-Phenyl-2-cyclohexene-1-alkylamine derivatives, process for their preparation and medicines containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-08-05 EP disclosed