SCHEMBL11078634

SCHEMBL11078634

CCCc1nc(C=O)c(C)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.38
POLB P06746 1/20 0.36
ALK Q9UM73 1/20 0.35
KDM4C Q9H3R0 1/20 0.34
ADORA2A P29274 3/20 0.33
ADORA1 P30542 3/20 0.33
ADORA3 P0DMS8 2/20 0.33
KDM4E B2RXH2 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK1 P28482 1/20 0.32
PARP1 P09874 1/20 0.32
CDK1 P06493 1/20 0.30
CCNB1 P14635 1/20 0.30
GPR84 Q9NQS5 1/20 0.30
PDE5A O76074 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2033187 0.84 ALK (0.46) ALKADORA2AADORA1ADORA3CDK1
SCHEMBL4352906 0.81 GLA (0.38) GLAPOLBKDM4CADORA2AADORA1
SCHEMBL7763940 0.79 GLA (0.37) GLAPOLBKDM4CADORA2AADORA1
SCHEMBL10802354 0.74 CYP1A2 (0.34) GLAPOLBKDM4EKMT2ACDK1
SCHEMBL10802364 0.74 CYP1A2 (0.34) GLAPOLBKDM4EKMT2ACDK1
SCHEMBL9308282 0.73 GLA (0.38) GLAPOLBKDM4CKDM4EKMT2A
SCHEMBL7369422 0.73 HSD17B10 (0.50) POLBKDM4EMAPK1
SCHEMBL3703329 0.73 GLA (0.40) GLAPOLBKDM4CADORA2AADORA1
SCHEMBL9138920 0.72 ADORA3 (0.33) GLAPOLBKDM4CADORA2AADORA1
SCHEMBL3701645 0.71 GLA (0.39) GLAPOLBKDM4CADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447603-A ANTI -ASTHMATICS AMERICAN CYANAMID COMPANY (US) 1984-05-08 US disclosed
EP-0057289-A1 1-Substituted-6-n-propyl-8-methylimidazo(1,5-d)-as-triazin-4(3H)-ones AMERICAN CYANAMID COMPANY (US) 1982-08-11 EP disclosed
US-RE30511-E ENZYME INHIBITOR, HERBICIDE, CYCLIZATION AMERICAN CYANAMID COMPANY (US) 1981-02-10 US disclosed
US-4168964-A HERBICIDES AMERICAN CYANAMID COMPANY (US) 1979-09-25 US disclosed
US-4124766-A INTERMEDIATES FOR PHOSPHODIESTERASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1978-11-07 US disclosed
US-4107308-A HYPOTENSIVE AGENTS, HERBICIDES, REACTING SODIUM SALT WITH ALLYL OR ALKYL HALIDE, RING CLOSURE AMERICAN CYANAMID COMPANY (US) 1978-08-15 US disclosed
US-4107307-A ENZYME INHIBITORS, HERBICIDES, RING CLOSURE AMERICAN CYANAMID COMPANY (US) 1978-08-15 US disclosed