SCHEMBL11080641

SCHEMBL11080641

COc1cc(C2(N(C)C)CCC(N(C)CCc3ccccc3)CC2)ccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
OPRM1 P35372 7/20 0.41
OPRL1 P41146 7/20 0.41
GRIN2B Q13224 2/20 0.40
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2A P28223 1/20 0.38
HTR1E P28566 1/20 0.38
HTR7 P34969 1/20 0.38
HTR2B P41595 1/20 0.38
HTR5A P47898 1/20 0.38
HTR6 P50406 1/20 0.38
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
HPGD P15428 1/20 0.36
SLC18A3 Q16572 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11071655 0.83 SLC6A4 (0.53) POLBOPRM1OPRL1SLC6A4SLC6A3
SCHEMBL11078301 0.82 OPRL1 (0.58) OPRM1OPRL1GRIN2B
SCHEMBL11066830 0.81 OPRL1 (0.46) OPRM1OPRL1GRIN2BSLC18A3
Ethylbenzene SCHEMBL11080651 0.78 OPRL1 (0.45) OPRM1OPRL1SLC6A4SLC6A3
SCHEMBL11065445 0.77 OPRM1 (0.58) OPRM1OPRL1GRIN2BSLC18A3
SCHEMBL11073158 0.77 OPRM1 (0.50) OPRM1OPRL1GRIN2B
SCHEMBL11079938 0.76 OPRL1 (0.46) OPRM1OPRL1GRIN2B
SCHEMBL11070020 0.75 OPRM1 (0.49) OPRM1OPRL1GRIN2B
SCHEMBL11077368 0.75 GRIN2B (0.42) OPRM1OPRL1GRIN2BSLC18A3
SCHEMBL11076128 0.74 CHIA (0.44) OPRM1OPRL1GRIN2BSLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447454-A Analgetic compounds, compositions and process of treatment THE UPJOHN COMPANY (US) 1984-05-08 US disclosed
US-4113866-A ANALGETIC COMPOUNDS, COMPOSITIONS AND PROCESS OF TREATMENT THE UPJOHN COMPANY (US) 1978-09-12 US disclosed