SCHEMBL11084683

SCHEMBL11084683

CC(C)(C)OC(=O)C1NCCN(CC(=O)O)C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 5/20 0.41
PLA2G10 O15496 2/20 0.35
PLA2G5 P39877 2/20 0.35
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPK1 P28482 1/20 0.31
STS P08842 1/20 0.31
KDM4E B2RXH2 2/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
RECQL P46063 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
ITGB3 P05106 1/20 0.30
ITGA2B P08514 1/20 0.30
PKM P14618 2/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7309781 0.85 ACE (0.44) ACELMNAPOLBCYP2D6CYP2C9
SCHEMBL7309788 0.85 ACE (0.44) ACELMNAPOLBCYP2D6CYP2C9
SCHEMBL18205531 0.82 PLA2G10 (0.34) PLA2G10PLA2G5MAPK1
SCHEMBL8988835 0.77 ACE (0.39) ACEPLA2G10PLA2G5LMNAPOLB
SCHEMBL8988818 0.77 ACE (0.39) ACEPLA2G10PLA2G5LMNAPOLB
SCHEMBL11092369 0.74 MMP13 (0.48) ACEKMT2AKDM4EALDH1A1
SCHEMBL8544676 0.74 MMP13 (0.44) POLBKMT2A
SCHEMBL18205336 0.74 PLA2G10 (0.32) PLA2G10PLA2G5MAPK1
SCHEMBL7309092 0.73 MEN1 (0.40) ACEKMT2ATDP1GAA
SCHEMBL7309103 0.73 MEN1 (0.40) ACEKMT2ATDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4483988-A Substituted derivatives of 4-t-alkoxycarbonyl-piperazin-2-ones RICHARDSON MERRELL INC. (US) 1984-11-20 US disclosed
US-4435571-A 5-(Substituted benzyl)-6-oxo-2-piperazine carboxylic acids and esters RICHARDSON MERRELL INC. (US) 1984-03-06 US disclosed
US-4341698-A Enkaphalin derivatives RICHARDSON-MERRELL INC. (US) 1982-07-27 US disclosed