SCHEMBL7309788

SCHEMBL7309788

COC(=O)C1NCCN(CC(=O)O)C1=O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACE P12821 5/20 0.44
LMNA P02545 1/20 0.35
FKBP1A P62942 2/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PKM P14618 2/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ITGB3 P05106 4/20 0.33
ITGA2B P08514 4/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
RECQL P46063 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7309781 1.00 ACE (0.44) ACELMNAFKBP1AKMT2APOLB
SCHEMBL11084683 0.85 ACE (0.41) ACELMNAKMT2APOLBCYP2D6
SCHEMBL7311432 0.77 PKM (0.45) ACELMNAPKMGAAITGB3
SCHEMBL7311444 0.77 PKM (0.45) ACELMNAPKMGAAITGB3
SCHEMBL8988835 0.71 ACE (0.39) ACELMNAKMT2APOLBCYP2D6
SCHEMBL8988818 0.71 ACE (0.39) ACELMNAKMT2APOLBCYP2D6
SCHEMBL691684 0.68 PKM (0.51) KMT2APKMGAAALDH1A1
Hydrochloric Acid SCHEMBL7277753 0.68 PKM (0.44) ACEKMT2APOLBCYP2D6CYP2C9
SCHEMBL7366324 0.68 PKM (0.44) KMT2APKMGAAITGB3ITGA2B
Hydrochloric Acid SCHEMBL7277734 0.68 PKM (0.44) ACEKMT2APOLBCYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643072-B1 2-Piperazinone compounds and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-02-24 EP disclosed
US-5550131-A ANTITHROMBOTIC AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-27 US disclosed
EP-0643072-A1 2-Piperazinone compounds and their use Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed