SCHEMBL1108637

SCHEMBL1108637

CNC1CN2CCC1CC2

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.48
CA1 P00915 3/20 0.48
CA2 P00918 3/20 0.48
CA9 Q16790 3/20 0.48
CHRNA7 P36544 4/20 0.42
GAA P10253 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
KAT2B Q92831 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13874664 1.00 CA12 (0.48) CA12CA1CA2CA9CHRNA7
SCHEMBL9431723 1.00 CA12 (0.48) CA12CA1CA2CA9CHRNA7
SCHEMBL15291340 1.00 CA12 (0.48) CA12CA1CA2CA9CHRNA7
SCHEMBL2823734 1.00 CA12 (0.48) CA12CA1CA2CA9CHRNA7
Hydrochloric Acid SCHEMBL492681 0.98 CA12 (0.47) CA12CA1CA2CA9CHRNA7
Hydrochloric Acid SCHEMBL493210 0.98 CA12 (0.47) CA12CA1CA2CA9CHRNA7
Hydrochloric Acid SCHEMBL9706304 0.98 CA12 (0.47) CA12CA1CA2CA9CHRNA7
SCHEMBL13624167 0.88
SCHEMBL8432427 0.75 CA12 (0.48) CA12CA1CA2CA9CHRNA7
SCHEMBL13146329 0.75 CA12 (0.48) CA12CA1CA2CA9CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 175 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250026749-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GENZYME CORPORATION (US) 2025-01-23 US disclosed
US-12060349-B2 Glucosylceramide synthase inhibitors GENZYME CORPORATION (US) 2024-08-13 US disclosed
WO-2023202735-A1 POLYMER CONJUGATE FOR BLOCKING OF NON-SPECIFIC INTERACTIONS IN IMMUNOCHEMICAL ASSAYS, METHOD OF ITS SYNTHESIS AND USE THEREOF USTAV MAKROMOLEKULARNI CHEMIE AV CR, V.V.I. (CZ) 2023-10-26 WO disclosed
US-20230301990-A1 CERTAIN ARYL PLADIENOLIDE COMPOUNDS AND METHODS OF USE EISAI R&D MANAGEMENT CO., LTD. (JP) 2023-09-28 US disclosed
US-20230301990-A1 CERTAIN ARYL PLADIENOLIDE COMPOUNDS AND METHODS OF USE EISAI R&D MANAGEMENT CO., LTD. (JP) 2023-09-28 US disclosed
US-20230203022-A1 HETEROCYCLE AND GLUTARIMIDE SKELETON-BASED COMPOUND AND APPLICATIONS THEREOF SHANGHAITECH UNIVERSITY (CN) 2023-06-29 US disclosed
US-11679107-B2 Certain aryl pladienolide compounds and methods of use EISAI R&D MANAGEMENT CO., LTD. (JP) 2023-06-20 US disclosed
US-11679107-B2 Certain aryl pladienolide compounds and methods of use EISAI R&D MANAGEMENT CO., LTD. (JP) 2023-06-20 US disclosed
EP-3724188-B1 PROGRANULIN MODULATORS AND METHODS OF USING THE SAME ARKUDA THERAPEUTICS (US) 2023-06-07 EP disclosed
EP-3724188-B1 PROGRANULIN MODULATORS AND METHODS OF USING THE SAME ARKUDA THERAPEUTICS (US) 2023-06-07 EP disclosed
EP-1548121-A1 NOVEL PHYSIOLOGICALLY ACTIVE SUBSTANCES MERCIAN CORPORATION (JP) 2005-06-29 EP disclosed
EP-1541570-A1 NOVEL PHYSIOLOGICALLY ACTIVE SUBSTANCE MERCIAN CORPORATION (JP) 2005-06-15 EP disclosed
EP-1508570-A1 NOVEL PHYSIOLGICALLY ACTIVE SUBSTANCES MERCIAN CORPORATION (JP) 2005-02-23 EP disclosed
WO-2004103998-A1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LIMITED (GB) 2004-12-02 WO disclosed
WO-2004024728-A2 PYRAZOLO[3,4-B]PYRIDINE COMPOUNDS, AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LIMITED (GB) 2004-03-25 WO disclosed
EP-0720601-B1 GASTRIN AND CCK RECEPTOR LIGANDS BLACK JAMES FOUNDATION (GB) 2000-10-25 EP disclosed
EP-0720601-A1 GASTRIN AND CCK RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 1996-07-10 EP disclosed
WO-1995004720-A2 GASTRIN AND CCK RECEPTOR LIGANDS BLACK JAMES FOUNDATION (GB) 1995-02-16 WO disclosed
US-5192770-A Antiemetic, anxiolytic, cognition activator SYNTEX (U.S.A.) INC. (US) 1993-03-09 US disclosed
EP-0490263-A1 Alpha-oxoacetamide derivatives SYNTEX (U.S.A.) INC. (US) 1992-06-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11679107-B2 Certain aryl pladienolide compounds and methods of use PLAAT5, PLAAT3, SNRPE CA12 4246/4885CA1 4808/4885CA2 4707/4885
US-20230301990-A1 CERTAIN ARYL PLADIENOLIDE COMPOUNDS AND METHODS OF USE PLAAT5, PLAAT3, PLAAT4 CA12 4287/4885CA1 4837/4885CA2 4773/4885
US-20230203022-A1 HETEROCYCLE AND GLUTARIMIDE SKELETON-BASED COMPOUND AND APPLICATIONS THEREOF TNF, GCDH, LITAF CA12 1702/4885CA1 1446/4885CA2 1246/4885
US-12060349-B2 Glucosylceramide synthase inhibitors GBA1, GBA2, GALC CA12 1083/4885CA1 1779/4885CA2 845/4885
US-20250026749-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GBA1, GBA2, GAA CA12 1744/4885CA1 3275/4885CA2 2213/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.