SCHEMBL11088974

SCHEMBL11088974

CCOC(=O)CCCCCCC(NC(CC(=O)C(C)(C)C)c1ccccc1)C(=O)OCC

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 1/20 0.40
ACE P12821 1/20 0.39
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
LTA4H P09960 1/20 0.38
NAMPT P43490 1/20 0.38
ALOX5 P09917 1/20 0.37
FAAH O00519 2/20 0.37
POLB P06746 1/20 0.37
MMP8 P22894 1/20 0.37
TOP2A P11388 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11088418 0.74 CYP3A4 (0.47) CYP3A4CYP2D6CYP2C19KMT2AALDH1A1
SCHEMBL711239 0.73 CYP3A4 (0.52) CYP3A4CYP2D6CYP2C19ALDH1A1CYP4F2
SCHEMBL11091798 0.73 ALDH1A1 (0.46) CYP3A4CYP2D6CYP2C19KMT2AALDH1A1
SCHEMBL11092690 0.73 KMT2A (0.50) CYP3A4CYP2C19KMT2AALDH1A1NAMPT
SCHEMBL11267493 0.71 ALOX5 (0.43) CYP3A4CYP2D6CYP2C19KMT2AALDH1A1
Bromide SCHEMBL11083780 0.71 ALOX5 (0.49) KMT2AALDH1A1CYP4F2CYP4A11LTA4H
SCHEMBL11396997 0.71 ALDH1A1 (0.45) CYP3A4CYP2D6CYP2C19KMT2AALDH1A1
SCHEMBL11095337 0.71 KMT2A (0.41) CYP3A4CYP2D6CYP2C19KMT2AALDH1A1
SCHEMBL11094819 0.70 ALDH1A1 (0.44) CYP3A4CYP2D6CYP2C19KMT2AALDH1A1
SCHEMBL11093116 0.69 ALDH1A1 (0.43) CYP3A4CYP2D6CYP2C19KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4486443-A PROSTAGLANDIN-LIKE EFFECTS BURROUGHS WELLCOME CO. (US) 1984-12-04 US disclosed
EP-0001238-B1 HYDANTOIN DERIVATIVES, THEIR SYNTHESIS, PHARMACEUTICAL FORMULATIONS AND INTERMEDIATES IN THEIR PREPARATION THE WELLCOME FOUNDATION LIMITED (GB) 1984-07-04 EP disclosed
US-4262128-A HAVING PROSTAGLANDIN-LIKE BIOLOGICAL PROPERTIES BURROUGHS WELLCOME CO. (US) 1981-04-14 US disclosed
US-4204068-A Nitrogen heterocycles BURROUGHS WELLCOME CO. (US) 1980-05-20 US disclosed
EP-0001238-A1 Hydantoin derivatives, their synthesis, pharmaceutical formulations and intermediates in their preparation THE WELLCOME FOUNDATION LIMITED (GB) 1979-04-04 EP disclosed