SCHEMBL11089031

SCHEMBL11089031

Cc1ccccc1Nc1noc(N)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.57
NPC1 O15118 4/20 0.53
RAB9A P51151 4/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
LMNA P02545 1/20 0.53
PKM P14618 1/20 0.53
NFKB1 P19838 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53
LRRK2 Q5S007 1/20 0.48
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 1/20 0.46
NPSR1 Q6W5P4 2/20 0.45
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
NTSR1 P30989 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
SLC2A1 P11166 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11089178 0.88 NPC1 (0.52) HTTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL11085839 0.81 TSHR (0.56) NPC1RAB9ASMN1; SMN2LMNALRRK2
SCHEMBL13750837 0.78 HTT (0.59) HTTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL23795778 0.78 NPC1 (0.71) HTTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL27628518 0.78 NPC1 (0.71) HTTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL17403482 0.76 MAPT (0.52) HTTNPC1RAB9ASMN1; SMN2PKM
SCHEMBL11086975 0.75 LMNA (0.57) RAB9ASMN1; SMN2LMNALRRK2ALDH1A1
SCHEMBL31261584 0.74 NPC1 (0.47) HTTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL20355153 0.74 HTT (0.69) HTTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL11088916 0.73 RAB9A (0.53) HTTNPC1RAB9ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4446142-A HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-05-01 US claimed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP claimed
US-4446142-A HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-05-01 US disclosed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP disclosed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP disclosed