SCHEMBL11088916

SCHEMBL11088916

Cc1ccc(Nc2noc(N)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.53
NPC1 O15118 6/20 0.47
JAK2 O60674 1/20 0.47
KCNH2 Q12809 1/20 0.45
SCN5A Q14524 1/20 0.45
SCN9A Q15858 1/20 0.45
SMN1; SMN2 Q16637 6/20 0.44
HTT P42858 2/20 0.44
TUBB4A P04350 2/20 0.44
TUBB P07437 2/20 0.44
TUBA3C P0DPH7 2/20 0.44
TUBA1B P68363 2/20 0.44
TUBA4A P68366 2/20 0.44
TUBB4B P68371 2/20 0.44
TUBB3 Q13509 2/20 0.44
TUBB2A Q13885 2/20 0.44
TUBB8 Q3ZCM7 2/20 0.44
TUBA3E Q6PEY2 2/20 0.44
TUBA1A Q71U36 2/20 0.44
TUBA1C Q9BQE3 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11089778 0.81 SMN1; SMN2 (0.53) RAB9ANPC1KCNH2SCN5ASCN9A
SCHEMBL11080475 0.81 MEN1 (0.53) RAB9ANPC1KCNH2SCN5ASCN9A
SCHEMBL17403482 0.81 MAPT (0.52) RAB9ANPC1SMN1; SMN2HTTCYP1A2
SCHEMBL19075472 0.79 RAB9A (0.51) RAB9ANPC1SMN1; SMN2TUBB4ATUBB
SCHEMBL12253181 0.75 NPC1 (0.61) RAB9ANPC1JAK2SMN1; SMN2HTT
SCHEMBL11078558 0.74 POLA1 (0.50) LMNATDO2NPY5RMAPK1
SCHEMBL11089031 0.73 HTT (0.57) RAB9ANPC1SMN1; SMN2HTTLMNA
SCHEMBL10938637 0.73 TUBB4A (0.58) RAB9ANPC1JAK2KCNH2SCN5A
SCHEMBL16014242 0.70 MAPT (0.44) GAAMAPTMEN1KMT2A
SCHEMBL20355151 0.70 RAB9A (0.67) RAB9ANPC1JAK2KCNH2SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4446142-A HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-05-01 US claimed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP claimed
US-4446142-A HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-05-01 US disclosed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP disclosed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP disclosed