SCHEMBL11089178

SCHEMBL11089178

Cc1cccc(Nc2noc(N)n2)c1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.52
RAB9A P51151 5/20 0.52
HTT P42858 3/20 0.52
JAK2 O60674 1/20 0.52
TNF P01375 1/20 0.52
NOD1 Q9Y239 1/20 0.52
NUDT1 P36639 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 3/20 0.44
TP53 P04637 1/20 0.44
RAPGEF4 Q8WZA2 1/20 0.44
LMNA P02545 3/20 0.42
NFKB1 P19838 2/20 0.42
NFKB2 Q00653 2/20 0.42
RELA Q04206 2/20 0.42
PKM P14618 2/20 0.42
CCR4 P51679 1/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
KDM4E B2RXH2 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11089031 0.88 HTT (0.57) NPC1RAB9AHTTSMN1; SMN2MAPT
SCHEMBL31453494 0.78 RAB9A (0.73) NPC1RAB9AHTTJAK2TNF
SCHEMBL11085839 0.73 TSHR (0.56) NPC1RAB9ASMN1; SMN2MAPTLMNA
SCHEMBL4189645 0.72 RAPGEF4 (0.65) NPC1RAB9ANUDT1SMN1; SMN2MAPT
SCHEMBL10410878 0.71 TSHR (0.58) NPC1RAB9AHTTJAK2TNF
SCHEMBL11403543 0.70 KMT2A (0.61) NPC1RAB9AHTTNUDT1SMN1; SMN2
SCHEMBL4544854 0.70 SLC2A1 (0.52) NPC1RAB9AHTTJAK2TNF
SCHEMBL11088916 0.69 RAB9A (0.53) NPC1RAB9AHTTJAK2SMN1; SMN2
SCHEMBL1922753 0.68 LMNA (0.63) NPC1RAB9AHTTNUDT1SMN1; SMN2
SCHEMBL17403482 0.68 MAPT (0.52) NPC1RAB9AHTTSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4446142-A HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-05-01 US claimed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP claimed
US-4446142-A HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-05-01 US disclosed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP disclosed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP disclosed