SCHEMBL11090448

SCHEMBL11090448

N=C(NC(N)=O)Nc1c(F)cccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.43
CYP1A2 P05177 1/20 0.43
KMT2A Q03164 2/20 0.41
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
TLR7 Q9NYK1 2/20 0.40
BACE1 P56817 1/20 0.40
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
PLAU P00749 1/20 0.38
PLAT P00750 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4098970 0.89 KMT2A (0.46) GAAKMT2AJAK2JAK1TYK2
Biclodil SCHEMBL1815631 0.89 CYP1A2 (0.49) CYP1A2KMT2ATYK2F2F10
SCHEMBL11274193 0.88 BACE1 (0.42) GAACYP1A2KMT2ATLR7BACE1
Biclodil SCHEMBL121552 0.87 CYP1A2 (0.47) CYP1A2KMT2ATYK2F2F10
SCHEMBL11089784 0.82 L3MBTL1 (0.47) CYP1A2TYK2POLBPTGS2
SCHEMBL11093150 0.82 CYP1A2 (0.43) CYP1A2KMT2ATYK2F2F10
SCHEMBL11582985 0.82 HTT (0.40) KMT2AJAK1TLR7CA12CA1
SCHEMBL11579586 0.82 DRD2 (0.44) CYP1A2KMT2AF2F10PLAU
SCHEMBL4099006 0.82 GAA (0.51) GAACYP1A2POLB
SCHEMBL11056409 0.82 KMT2A (0.47) GAACYP1A2KMT2AJAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4446152-A SUBSTITUTED PHENYLAMIDINOUREA WILLIAM H. RORER, INC. (US) 1984-05-01 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed