SCHEMBL11089784

SCHEMBL11089784

N=C(NC(N)=O)Nc1c(Cl)cccc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.47
PTGS2 P35354 1/20 0.45
TYK2 P29597 1/20 0.45
GBA1 P04062 1/20 0.42
HPGD P15428 1/20 0.41
PDK1 Q15118 2/20 0.41
PDK2 Q15119 2/20 0.41
PDK3 Q15120 2/20 0.41
PDK4 Q16654 2/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KLK1 P06870 1/20 0.39
KLK5 Q9Y337 1/20 0.39
CLCN2 P51788 1/20 0.39
KCNJ5 P48544 1/20 0.38
KCNJ3 P48549 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biclodil SCHEMBL1815631 0.86 CYP1A2 (0.49) TYK2PDK1PDK2PDK3PDK4
SCHEMBL11583003 0.86 PTGS2 (0.43) PTGS2
Biclodil SCHEMBL121552 0.85 CYP1A2 (0.47) TYK2PDK1PDK2PDK3PDK4
SCHEMBL11578713 0.84 SMN1; SMN2 (0.42) L3MBTL1TYK2LMNA
SCHEMBL11578620 0.84 RIPK1 (0.42) L3MBTL1HPGDPDK1PDK2PDK3
SCHEMBL11431335 0.83 L3MBTL1 (0.47) L3MBTL1PTGS2TYK2GBA1HPGD
SCHEMBL11090448 0.82 GAA (0.43) PTGS2TYK2CYP1A2POLB
SCHEMBL11884358 0.82 L3MBTL1 (0.47) L3MBTL1PTGS2TYK2GBA1HPGD
SCHEMBL11579856 0.81 MAPK1 (0.47) L3MBTL1PTGS2TYK2GBA1HPGD
SCHEMBL11579402 0.80 ALDH1A1 (0.43) PDK1PDK2PDK3PDK4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4446152-A SUBSTITUTED PHENYLAMIDINOUREA WILLIAM H. RORER, INC. (US) 1984-05-01 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed