SCHEMBL11093075

SCHEMBL11093075

COC(=O)C(Cc1ccccc1)N1CN(C(Cc2ccccc2)C(=O)OC)CN(C(Cc2ccccc2)C(=O)OC)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
ATM Q13315 1/20 0.48
LMNA P02545 1/20 0.48
CYP2C9 P11712 3/20 0.47
CYP2C19 P33261 3/20 0.47
HSD17B10 Q99714 3/20 0.47
POLB P06746 3/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
RECQL P46063 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
PTPN7 P35236 1/20 0.47
BLM P54132 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
GFER P55789 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11095987 0.88 LTA4H (0.61) NPC1RAB9A
SCHEMBL3191795 0.88 NPC1 (0.46) NPC1RAB9AATMLMNACYP2C9
SCHEMBL3191801 0.88 NPC1 (0.46) NPC1RAB9AATMLMNACYP2C9
SCHEMBL1683002 0.86 RAB9A (0.58) NPC1RAB9AATMLMNACYP2C9
SCHEMBL19037806 0.84 LMNA (0.49) NPC1RAB9AATMLMNACYP2C9
SCHEMBL17294909 0.82 GAA (0.44) NPC1RAB9AATMLMNACYP2C9
SCHEMBL17294908 0.82 GAA (0.44) NPC1RAB9AATMLMNACYP2C9
SCHEMBL17304924 0.82 GAA (0.44) NPC1RAB9AATMLMNACYP2C9
SCHEMBL16984754 0.81 NPSR1 (0.68) RAB9AHSD17B10POLBKMT2AMEN1
SCHEMBL9650037 0.80 ALDH1A1 (0.70) NPC1RAB9AATMCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4483988-A Substituted derivatives of 4-t-alkoxycarbonyl-piperazin-2-ones RICHARDSON MERRELL INC. (US) 1984-11-20 US disclosed
US-4341698-A Enkaphalin derivatives RICHARDSON-MERRELL INC. (US) 1982-07-27 US disclosed