SCHEMBL11093239

SCHEMBL11093239

COC(=O)C(C)CC(C#N)(CCC(=O)O)c1ccccc1Cl

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
ESRRB O95718 1/20 0.33
NOS3 P29474 3/20 0.32
NOS1 P29475 3/20 0.32
NOS2 P35228 3/20 0.32
ANPEP P15144 3/20 0.32
ADRB2 P07550 2/20 0.32
ADRB1 P08588 2/20 0.32
ADRB3 P13945 2/20 0.32
HTT P42858 1/20 0.32
PTGFR P43088 3/20 0.32
NPC1 O15118 1/20 0.32
CNR1 P21554 1/20 0.32
CASP3 P42574 1/20 0.32
CASP6 P55212 1/20 0.32
CASP8 Q14790 1/20 0.32
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11823083 0.91 CYP2C9 (0.31) ALDH1A1ADRB3CNR1CASP3CASP6
SCHEMBL11821438 0.85 ESRRB (0.36) ALDH1A1ESRRBANPEPKMT2A
SCHEMBL11821434 0.85 CYP1A2 (0.35) ALDH1A1ESRRBADRB2ADRB1ADRB3
SCHEMBL11817919 0.82 GRIN2D (0.39) ALDH1A1NOS3NOS1NOS2CNR1
SCHEMBL11097563 0.82 FFAR1 (0.38) ALDH1A1HTTPTGFRKMT2A
SCHEMBL11826141 0.78 MEN1 (0.32) ALDH1A1KMT2A
SCHEMBL11097440 0.78 CTSC (0.33) ALDH1A1ESRRBANPEPNPC1KMT2A
SCHEMBL11823939 0.78 ALDH1A1 (0.38) ALDH1A1HTTKMT2A
SCHEMBL11821704 0.77 KIF11 (0.39) ALDH1A1HTTNPC1
SCHEMBL11821371 0.77 CTSL (0.38) ALDH1A1NOS3NOS1NOS2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed