SCHEMBL11095484

SCHEMBL11095484

CCCCCCN1C2CCC1CC(C(=O)Nc1cc(Cl)c(N)cc1OC)C2

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 5/20 0.52
TSHR P16473 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
ACHE P22303 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11100115 0.88 TSHR (0.45) HTR4TSHRMEN1ALDH1A1KMT2A
SCHEMBL11100788 0.86 TSHR (0.43) HTR4TSHRMEN1ALDH1A1KMT2A
SCHEMBL11278608 0.85 HTR4 (0.48) HTR4TSHR
SCHEMBL11095690 0.85 KMT2A (0.51) MEN1ALDH1A1KMT2A
SCHEMBL11098785 0.85 CHEK1 (0.41) HTR4TSHRMEN1ALDH1A1KMT2A
SCHEMBL11096503 0.83 DRD2 (0.52) HTR4CYP2D6CYP2C9ACHE
SCHEMBL11094874 0.82 DRD2 (0.61) CYP2D6CYP2C9ACHE
SCHEMBL11099827 0.82 TSHR (0.49) HTR4TSHRACHE
SCHEMBL11092428 0.82 DRD2 (0.52) HTR4TSHR
SCHEMBL11097949 0.81 DRD2 (0.51) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0031219-B1 ANILINE DERIVATIVES BEECHAM GROUP PLC (GB) 1984-03-07 EP disclosed
US-4350691-A ANTIEMETICS BEECHAM GROUP LIMITED (GB) 1982-09-21 US disclosed
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP disclosed