SCHEMBL11100788

SCHEMBL11100788

CCCCCCN1C2CCC1CC(C(=O)Nc1cc(Cl)c(NC=O)cc1OC)C2

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.43
TMEM97 Q5BJF2 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HTR4 Q13639 2/20 0.38
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
DRD4 P21917 4/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11100115 0.89 TSHR (0.45) TSHRTMEM97SIGMAR1ALDH1A1LMNA
SCHEMBL11099467 0.86 TSHR (0.44) TSHRKMT2AMEN1DRD4
SCHEMBL11095484 0.86 HTR4 (0.52) TSHRALDH1A1HTR4KMT2AMEN1
SCHEMBL11096161 0.84 DRD4 (0.51) TSHROPRM1OPRD1DRD4SMN1; SMN2
SCHEMBL11095690 0.83 KMT2A (0.51) TMEM97SIGMAR1ALDH1A1NPSR1KMT2A
SCHEMBL11098785 0.83 CHEK1 (0.41) TSHRTMEM97SIGMAR1ALDH1A1LMNA
SCHEMBL11093528 0.83 CXCR6 (0.47) TSHRSIGMAR1NPSR1DRD4
SCHEMBL11096423 0.83 TSHR (0.49) TSHRALDH1A1LMNAL3MBTL1OPRM1
SCHEMBL11097324 0.83 DRD4 (0.48) TSHROPRM1DRD4
SCHEMBL11094396 0.82 SIGMAR1 (0.46) TSHRSIGMAR1OPRM1OPRD1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0031219-B1 ANILINE DERIVATIVES BEECHAM GROUP PLC (GB) 1984-03-07 EP disclosed
US-4350691-A ANTIEMETICS BEECHAM GROUP LIMITED (GB) 1982-09-21 US disclosed
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP disclosed