SCHEMBL11096193

SCHEMBL11096193

CC(Oc1ccc(N(C)c2nnc3cc(Cl)ccc3n2)cc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.42
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
ALOX15 P16050 1/20 0.42
NFKB1 P19838 1/20 0.42
HIF1A Q16665 1/20 0.42
GMNN O75496 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
APEX1 P27695 1/20 0.42
PMP22 Q01453 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAP4K4 O95819 2/20 0.41
TSHR P16473 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11097512 0.89 MAPT (0.46) CYP1A2ALDH1A1SMN1; SMN2TP53CYP3A4
SCHEMBL11098428 0.89 MAPT (0.55) CYP1A2ALDH1A1SMN1; SMN2TP53CYP3A4
SCHEMBL11097303 0.88 EPHX2 (0.42) CYP1A2ALDH1A1SMN1; SMN2TP53CYP3A4
SCHEMBL11097501 0.87 TDP1 (0.39) CYP1A2SMN1; SMN2TP53LMNAMAP4K4
SCHEMBL11095436 0.86 TDP1 (0.41) CYP1A2ALDH1A1SMN1; SMN2TP53CYP3A4
SCHEMBL11124251 0.85 PPARA (0.46) PTGDR2
SCHEMBL10733255 0.84 MAP4K4 (0.45) CYP1A2ALDH1A1SMN1; SMN2TP53CYP3A4
SCHEMBL10963800 0.83 MAP4K4 (0.42) CYP1A2ALDH1A1SMN1; SMN2TP53CYP3A4
SCHEMBL11264919 0.82 CYP1A2 (0.51) CYP1A2ALDH1A1SMN1; SMN2TP53CYP3A4
SCHEMBL11272939 0.81 CYP1A2 (0.39) CYP1A2ALDH1A1SMN1; SMN2TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024931-B1 1,2,4-BENZOTRIAZINYLAMINOPHENOXYALKANE CARBOXYLIC ACID DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES ICI AUSTRALIA LIMITED (AU) 1984-10-17 EP claimed
US-4310347-A Herbicidal 1,2,4-benzotriazines ICI AUSTRALIA LIMITED (AU) 1982-01-12 US claimed
EP-0024931-A2 1,2,4-Benzotriazinylaminophenoxyalkane carboxylic acid derivatives, processes for their preparation and their use as herbicides ICI AUSTRALIA LIMITED (AU) 1981-03-11 EP claimed
EP-0024931-B1 1,2,4-BENZOTRIAZINYLAMINOPHENOXYALKANE CARBOXYLIC ACID DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES ICI AUSTRALIA LIMITED (AU) 1984-10-17 EP disclosed
US-4310347-A Herbicidal 1,2,4-benzotriazines ICI AUSTRALIA LIMITED (AU) 1982-01-12 US disclosed
EP-0024931-A2 1,2,4-Benzotriazinylaminophenoxyalkane carboxylic acid derivatives, processes for their preparation and their use as herbicides ICI AUSTRALIA LIMITED (AU) 1981-03-11 EP disclosed