SCHEMBL11096932

SCHEMBL11096932

COc1cc(C(=O)CN2CCC(N3Cc4ccccc4OC3=O)CC2)cc(OC)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
GAA P10253 1/20 0.49
HTT P42858 2/20 0.45
TAAR1 Q96RJ0 1/20 0.45
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
PLD2 O14939 1/20 0.41
PLD1 Q13393 1/20 0.41
SCN1A P35498 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
FKBP1A P62942 2/20 0.40
SIGMAR1 Q99720 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MCHR1 Q99705 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11100292 0.91 ALDH1A1 (0.46) ALDH1A1GAAHTTPOLBMAPT
SCHEMBL11096821 0.83 SCN1A (0.47) POLBMAPTSCN1ASCN5ASCN9A
SCHEMBL11097138 0.79 MAOB (0.54) ALDH1A1HTTTAAR1MAPTMEN1
SCHEMBL11493471 0.76 SIGMAR1 (0.48) POLBSIGMAR1LMNA
SCHEMBL11101000 0.75 ALDH1A1 (0.41) ALDH1A1GAAMAPTSCN1ASCN5A
SCHEMBL11099575 0.73 CHRM4 (0.48) ALDH1A1POLBMAPTSCN1ASCN5A
SCHEMBL11180233 0.72 ALDH1A1 (0.45) ALDH1A1GAAHTTPOLBMAPT
SCHEMBL11031363 0.72 PLD2 (0.73) ALDH1A1PLD2PLD1KDM4ELMNA
SCHEMBL11096272 0.71 CHRM2 (0.54) SIGMAR1
SCHEMBL11099931 0.70 ALDH1A1 (0.38) ALDH1A1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0029707-B1 NOVEL PIPERIDINE DERIVATIVES, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM KYOWA HAKKO KOGYO CO., LTD (JP) 1984-02-01 EP disclosed
US-4390536-A HYPOTENSIVE AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1983-06-28 US disclosed
US-4344945-A HYPOTENSIVE AGENTS, BENZOXAZINYL DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1982-08-17 US disclosed
EP-0029707-A1 Novel piperidine derivatives, method for the preparation thereof and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1981-06-03 EP disclosed